Synthesis and Antibacterial Activity of Some Novel 1,4- Diazepines from β-Diketones/ β -Ketoesters of 4- Acetylaminobenzene Sulphonyl Chloride
نویسندگان
چکیده
A series of novel 1,4diazepines have been synthesized from β-diketones / β-ketoesters of 4acetylaminobenzene sulphonyl chloride. Desired compounds were prepared by the reaction of novel βdiketone / β-ketoester derivatives of [N4-(4acetylamino) benzene sulphonyl piperazinylN1-1bromopropane] with ethylenediamine to get 1, 4dizapines. All the newly synthesized compounds were characterized with IR and 1H NMR studies. Keywordsβ-diketone, β-ketoester, diazepines, ethylenediamine, antibacterial activities
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